Applying a Decade of Topoisomerase ADC Experience to Build the Next Generation of Payloads

  • Distil the most important translational and clinical lessons from the widespread adoption of topoisomerase I payloads across multiple tumor settings
  • Analyze which resistance mechanisms could have been anticipated and which only emerged through large-scale clinical use, informing more effective development strategies moving forward
  • Translate real-world experience into actionable guidance for designing nextgeneration topo payloads and identifying orthogonal mechanisms capable of addressing resistant patient populations